casein kinase — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T10687	Casein Kinase II Inhibitor IV		Casein Kinase
	Casein Kinase II Inhibitor IV is an inducer of epidermal keratinocyte differentiation.		Casein Kinase
T64350	Casein kinase 1δ-IN-3		Casein Kinase
	Casein kinase 1δ-IN-3 (Casein kinase 1δ-IN-3) (Compound 23a) is a casein kinase 1 delta (CK1d) inhibitor with a pIC50 of 6.5376 M.		Casein Kinase
T64376	Casein kinase 1δ-IN-9		NADPH
	Casein kinase 1δ-IN-9 is a Quinone reductase 2 inhibitor with IC50 of 0.6μM.		NADPH
T77500	Casein kinase 1δ-IN-6		Casein Kinase
	Casein kinase 1δ-IN-6 is a potent and selective inhibitor of the protein kinase CK-1δ with an IC50 of 23 nM.Casein kinase 1δ-IN-6 shows neuroprotective and anti-inflammatory activity in both in vitro and in vivo assays.C...		Casein Kinase
T9175	Casein Kinase inhibitor A51		Apoptosis , Casein Kinase
	Casein Kinase inhibitor A51 is an orally active casein kinase 1α (CK1α) inhibitor with anticancer activity that induces apoptosis in leukemia cells, and may be used in the study of neck cancers, acute myeloid leukemia, b...		Apoptosis , Casein Kinase
T60295	Casein kinase 1δ-IN-1	WAY-643895	Casein Kinase
	Casein kinase 1δ-IN-1 (WAY-643895) is an inhibitor of casein kinase 1δ (CK1δ), which inhibits CK1δ. Casein kinase 1δ-IN-1 can be used in the study of neurodegenerative diseases such as Alzheimer's disease.		Casein Kinase
T77648	Casein kinase 1δ-IN-14	WAY-637081	Others
	Casein kinase 1δ-IN-14 (WAY-637081) can be used to study atherosclerosis-related cardiovascular disease.		Others
T39482	Casein Kinase inhibitor A86	Casein Kinase inhibitor A86
	Casein Kinase inhibitor A86 is a highly effective and orally bioavailable inhibitor of casein kinase 1α (CK1α). Additionally, it displays inhibitory actions towards CDK7 (TFIIH) and CDK9 (P-TEFb). Furthermore, Casein Kin...
T77708	Casein kinase 1δ-IN-7		Casein Kinase
	Casein kinase 1δ-IN-7 is a Casein kinase 1δ inhibitor for neurodegenerative diseases such as Alzheimer's disease.		Casein Kinase
T77709	Casein kinase 1δ-IN-8		Casein Kinase
	Casein kinase 1δ-IN-8 is an inhibitor of casein kinase 1δ and is used to treat neurodegenerative diseases such as Alzheimer's disease type.		Casein Kinase
TP1509	Casein Kinase Substrates 3
	Casein Kinase Substrates 3 is a substrate of casein kinase.
T21915	TBCA	Casein Kinase II Inhibitor III, TBCA	Casein Kinase
	TBCA (Casein Kinase II Inhibitor III, TBCA) is a highly selective CK2 (casein kinase II) inhibitor, IC50 = 110 nM, Ki = 77 nM. TBCA shows selectivity for CK2 over CK1, DYRK1A and a panel of 27 other kinases.		Casein Kinase
T2449	D4476	D 4476,Casein Kinase I Inhibitor	Apoptosis , Casein Kinase , ALK , Autophagy
	D4476 (Casein Kinase I Inhibitor) is an effective, selective, and cell-permeant CK1 (casein kinase 1) inhibitor( IC50=300 nM in a cell-free assay).		Apoptosis , Casein Kinase , ALK , Autophagy
T7390	DMAT	Casein kinase II Inhibitor,CK2 Inhibitor	Casein Kinase
	DMAT (Casein kinase II Inhibitor) is a potent and specific inhibitor of CK2(IC50 value of 130 nM).		Casein Kinase
T2695	TBB	Casein Kinase II Inhibitor I,NSC 231634,4,5,6,7-tetrabromobenzotriazole	GSK-3 , Casein Kinase , CDK
	TBB (NSC-231634)(NSC-231634) is a highly selective, ATP/GTP-competitive inhibitor of casein kinase-2 (CK2).		GSK-3 , Casein Kinase , CDK
T10687L	Casein Kinase II Inhibitor IV Hydrochloride	Casein Kinase II Inhibitor IV Hydrochloride (863598-09-8 free base)	Others
	Casein Kinase II Inhibitor IV Hydrochloride is a small-molecule inducer of epidermal keratinocyte differentiation that lead to novel therapeutic approaches for the treatment of skin hyperproliferative disorders.		Others
T5358	Longdaysin		ERK , Casein Kinase , CDK
	Longdaysin is an inhibitor of CK1α and CK1δ (IC50s: 5.6/8.8 µM). It also can inhibit ERK2 (IC50: 52 µM).		ERK , Casein Kinase , CDK
T14069	A-3 hydrochloride		CaMK , Casein Kinase , PKA , PKC
	A-3 hydrochloride is a potent, cell-permeable, reversible, ATP-competitive non-selective antagonist of various kinases. A-3 hydrochloride also inhibits PKC and casein kinase I with Ki values of 47 µM and 80 µM, respectiv...		CaMK , Casein Kinase , PKA , PKC
T7949	NCC007		Casein Kinase
	NCC007 is a novel CKIα and CKIδ dual inhibitors by structural modification of N9 and C2 position of longdaysin.		Casein Kinase
T5056	PF-4800567		Casein Kinase
	PF-4800567 is a selective inhibitor of casein kinase 1ε (CK1ε; IC50 = 32 nM) with greater than 20-fold selectivity over CK1δ.		Casein Kinase